Azilsartan KaMedoxoMil CAS#863031-24-7

Azilsartan KaMedoxoMil CAS#863031-24-7

Azilsartan Kamedoxomil CAS#863031-24-7 yog angiotensin II receptor blocker. Azilsartan kamedoxomil yog ib qho organic potassium ntsev uas yog monopotassium ntsev ntawm azilsartan medoxomil. Ib tug prodrug rau azilsartan, nws yog siv rau kev kho mob ntshav siab.
Xa kev nug
Hauj lwm lawm
Product Description

 

Azilsartan Kamedoxomil CAS#863031-24-7 yog angiotensin II receptor blocker. Azilsartan kamedoxomil yog ib qho organic potassium ntsev uas yog monopotassium ntsev ntawm azilsartan medoxomil. Ib tug prodrug rau azilsartan, nws yog siv rau kev kho mob ntshav siab. Nws muaj lub luag haujlwm ua prodrug, tus neeg sawv cev tiv thaiv ntshav siab thiab angiotensin receptor antagonist. Nws muaj azilsartan medoxomil (1-).

Azilsartan kamedoxomil CAS#863031-24-7, tsim los ntawm Takeda Pharmaceuticals, tau pom zoo rau kev kho mob ntshav siab thiab tau tsim tawm hauv Asmeskas raws li lub npe Edarbi. Edarbi yog ib qho tshuaj uas ua rau muaj kev kub ntxhov ceev kom tso tawm azilsartan, cov khoom xyaw nquag (TAK-536, 39). Raws li 8th angiotensin receptor blocker (ARB) nkag mus rau hauv lub ntiaj teb ua lag luam, azilsartan kamedoxomil tuaj yeem ua haujlwm raws li kev kho mob monotherapy lossis ua ke nrog lwm cov tshuaj tiv thaiv kab mob. Hauv ntau qhov kev tshawb fawb soj ntsuam, monotherapeutic azilsartan kamedoxomil tau pom tias muaj kev tiv thaiv kab mob siab tshaj plaws thiab muaj txiaj ntsig zoo rau kev nyab xeeb / kev tiv thaiv kab mob hauv cov neeg mob piv nrog lwm cov kws kho mob, suav nrog valsartan, olmesartan medoxomil, candesartan, thiab telmisartan. -dose ua ke ntsiav tshuaj ntawm azilsartan kamedoxomil nrog chlorthalidone nyob rau hauv lub npe lag luam ntawm Edarbyclor.

 

Azilsartan kaMedoxoMil Chemical Properties

 

Melting point

193-195 degree

Cia temp.

Lub tub yees, nyob rau hauv inert cua

Solubility

DMSO (me ntsis), Methanol (me ntsis)

Daim ntawv

Khoom

Xim

Dawb rau Off-White

 

Cim npe nrov: azilsartan kamedoxomil cas#863031-24-7, Tuam Tshoj azilsartan kamedoxomil cas#863031-24-7 manufacturers, lwm tus neeg